Compile Data Set for Download or QSAR
maximum 50k data
Found 17 of ic50 data for polymerid = 50004466
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50302828(2-(4-(4-(butylcarbamoyl)-2-(2,4-dichlorophenylsulf...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]-PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362167(CHEMBL1941129)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362166(CHEMBL1941128)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50312906(2-(2-(bis(4-fluorophenyl)methyl)-4-(3-fluorophenyl...)
Affinity DataIC50:  29nMAssay Description:Inhibition of guinea pig CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362165(CHEMBL1941127)
Affinity DataIC50:  52nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50344991(2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl...)
Affinity DataIC50:  63nMAssay Description:Binding affinity to guinea pig CRTh2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362164(CHEMBL1941126)
Affinity DataIC50:  99nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362162(CHEMBL1941123)
Affinity DataIC50:  128nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362156(CHEMBL1941117)
Affinity DataIC50:  147nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362160(CHEMBL1941121)
Affinity DataIC50:  211nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362155(CHEMBL1941116)
Affinity DataIC50:  256nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362157(CHEMBL1941118)
Affinity DataIC50:  359nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362159(CHEMBL1941120)
Affinity DataIC50:  772nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362161(CHEMBL1941122)
Affinity DataIC50:  797nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362163(CHEMBL1941124)
Affinity DataIC50:  990nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362158(CHEMBL1941119)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50362168(CHEMBL1941125)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed